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a(SCHEM:"D-Glucose, anhydrous") -| path(SDIS:"muscle insulin receptor signaling pathway")
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Approximately 61,000 statements.
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Copyright (c) 2011-2012, Selventa. All rights reserved.
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Protein kinase C (PKC) is a serine kinase that has a number of potential substrates, including the insulin receptor (152). PKC is activated by the intracellular metabolite diacylglycerol (DAG), the concentration of which increases in a glucose-dependent manner during exposure of isolated muscles to hyperinsulinemia (153). In NIH3T3 cells overexpressing the insulin receptor, insulin desensitization by glucose can be blocked by PKC inhibitors and thiazolidinediones (154).
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